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Tukysa (tucatinib) is a small molecule pharmaceutical. Tucatinib was first approved as Tukysa on 2020-04-17. It is used to treat breast neoplasms in the USA. It has been approved in Europe to treat breast neoplasms and neoplasm metastasis. The pharmaceutical is active against receptor tyrosine-protein kinase erbB-2 and receptor tyrosine-protein kinase erbB-3. In addition, it is known to target epidermal growth factor receptor and receptor tyrosine-protein kinase erbB-4. Tukysa's patents are valid until 2032-10-12 (FDA).
Trade Name Tukysa
Common Name Tucatinib
Indication breast neoplasms, neoplasm metastasis
Drug Class Tyrosine kinase inhibitors
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