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Rapamune (sirolimus) is a small molecule pharmaceutical. Sirolimus was first approved as Rapamune on 1999-09-15. It has been approved in Europe to treat graft rejection and kidney transplantation. It is known to target peptidyl-prolyl cis-trans isomerase FKBP1A and peptidyl-prolyl cis-trans isomerase FKBP35.
Trade Name Rapamune
Common Name Sirolimus
Indication graft rejection, kidney transplantation
Drug Class Immunosuppressives: immunosuppressant, rapamycin derivatives
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