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Ponatinib

Iclusig (ponatinib) is a small molecule pharmaceutical. Ponatinib was first approved as Iclusig on 2012-12-14. It is used to treat myeloid leukemia in the USA. It has been approved in Europe to treat lymphoid leukemia and myeloid leukemia. The pharmaceutical is active against tyrosine-protein kinase ABL1. In addition, it is known to target cyclin-dependent kinase 19, proto-oncogene tyrosine-protein kinase receptor Ret, cyclin-dependent kinase 8, receptor-interacting serine/threonine-protein kinase 3, receptor-interacting serine/threonine-protein kinase 2, and receptor-interacting serine/threonine-protein kinase 1. Iclusig's patents are valid until 2033-12-12 (FDA).
Trade Name Iclusig
Common Name Ponatinib
Indication lymphoid leukemia, myeloid leukemia
Drug Class Tyrosine kinase inhibitors
Ponatinib
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