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Pexacerfont
Pexacerfont is a small molecule pharmaceutical. It is currently being investigated in clinical studies. It is known to target CRHR1-IT1-CRHR1 protein.
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Commercial
Therapeutic Areas
No data
Trade Name
FDA
EMA
No data
Drug Products
FDA
EMA
New Drug Application (NDA)
New Drug Application (NDA)
Abbreviated New Drug Application (ANDA)
Abbreviated New Drug Application (ANDA)
No data
Labels
FDA
EMA
No data
Indications
FDA
EMA
No data
Agency Specific
FDA
EMA
No data
Patent Expiration
No data
ATC Codes
No data
HCPCS
No data
Clinical
Clinical Trials
5 clinical trials
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Mock data
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Indications Phases 4
No data
Indications Phases 3
Indication
MeSH
Ontology
ICD-10
Ph 1
Ph 2
Ph 3
Ph 4
Other
Total
Anxiety disordersD001008EFO_0006788F41.1—21——2
Indications Phases 2
Indication
MeSH
Ontology
ICD-10
Ph 1
Ph 2
Ph 3
Ph 4
Other
Total
AlcoholismD000437EFO_0003829F10.1—1———1
Alcohol-related disordersD019973F10—1———1
Major depressive disorderD003865EFO_0003761F2211———1
Irritable bowel syndromeD043183EFO_0000555K58—1———1
Indications Phases 1
Indication
MeSH
Ontology
ICD-10
Ph 1
Ph 2
Ph 3
Ph 4
Other
Total
PlacebosD0109191————1
Indications Without Phase
No data
Epidemiology
Epidemiological information for investigational and approved indications
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Drug
General
Drug common namePEXACERFONT
INNpexacerfont
Description
Pexacerfont is a pyrazolopyridine.
Classification
Small molecule
Drug classCRF-1 (corticotropin releasing factor) receptor antagonists
Image (chem structure or protein)
Structure (InChI/SMILES or Protein Sequence)
CC[C@@H](C)Nc1nc(C)nc2c(-c3ccc(OC)nc3C)c(C)nn12
Identifiers
PDB—
CAS-ID459856-18-9
RxCUI—
ChEMBL IDCHEMBL482950
ChEBI ID—
PubChem CID9884366
DrugBankDB12572
UNII IDLF1VBG4ZUK (ChemIDplus, GSRS)
Target
Agency Approved
No data
Alternate
LINC02210-CRHR1
LINC02210-CRHR1
Organism
Homo sapiens
Gene name
LINC02210-CRHR1
Gene synonyms
CRFR, CRFR1, CRHR
NCBI Gene ID
104909134
Protein name
CRHR1-IT1-CRHR1 protein
Protein synonyms
Corticotropin-releasing hormone receptor 1, CRH-R-1, CRH-R1, CRHR1-IT1-CRHR1 readthrough
Uniprot ID
P34998
Mouse ortholog
—
—
Variants
Clinical Variant
No data
Financial
No data
Trends
PubMed Central
Top Terms for Disease or Syndrome:
Mock data
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Additional graphs summarizing 139 documents
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Safety
Black-box Warning
No Black-box warning
Adverse Events
Top Adverse Reactions
0 adverse events reported
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