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Hexylcaine
Cyclaine (hexylcaine) is a small molecule pharmaceutical. Hexylcaine was first approved as Cyclaine on 1982-01-01.
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Commercial
Therapeutic Areas
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Trade Name
FDA
EMA
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Drug Products
FDA
EMA
New Drug Application (NDA)
New Drug Application (NDA)
Abbreviated New Drug Application (ANDA)
Abbreviated New Drug Application (ANDA)
Hexylcaine hydrochloride
Tradename
Company
Number
Date
Products
CYCLAINEMerck KGaAN-008472 DISCN1982-01-01
1 products
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Labels
FDA
EMA
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Indications
FDA
EMA
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Agency Specific
FDA
EMA
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Patent Expiration
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ATC Codes
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HCPCS
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Clinical
Indications Phases 4
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Indications Phases 3
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Indications Phases 2
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Indications Phases 1
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Indications Without Phase
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Epidemiology
Epidemiological information for investigational and approved indications
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Drug
General
Drug common nameHEXYLCAINE
INNhexylcaine
Description
Hexylcaine hydrochloride, also called cyclaine (Merck) or osmocaine, is a short-acting local anesthetic. It acts by inhibiting sodium channel conduction. Overdose can lead to headache, tinnitus, numbness and tingling around the mouth and tongue, convulsions, inability to breathe, and decreased heart function.
Classification
Small molecule
Drug classlocal anesthetics
Image (chem structure or protein)
Structure (InChI/SMILES or Protein Sequence)
CC(CNC1CCCCC1)OC(=O)c1ccccc1
Identifiers
PDB
CAS-ID532-77-4
RxCUI26879
ChEMBL IDCHEMBL1197
ChEBI ID34791
PubChem CID10770
DrugBankDB00473
UNII ID511IU0826Z (ChemIDplus, GSRS)
Target
Agency Approved
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Alternate
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Variants
Clinical Variant
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Financial
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Trends
PubMed Central
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Safety
Black-box Warning
No Black-box warning
Adverse Events
Top Adverse Reactions
0 adverse events reported
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